Publications
2025
- Sustainable Copper-Catalyzed Cyanation of Aryl Iodine through a Design of Experiment Strategy
Brugemann K., Steinsoultz P. , Pereira T., Peter C., Hammoud S., Schmitt M., Blond G., Bihel F.
ACS Sustainable Chemistry & Engineering 2025, 10.1021/acssuschemeng.5c04898. - Double-Click Strategy Combining CuAAC and (Thia-) Diels-Alder Reactions; Application towards Peptide Labeling
Maujean T., Van Wesemael C., Tual L., Le Berruyer V., Rodriguez-Noguer B., Girard N., Bonnet D., Gulea M.
Chem. Eur. J. 2025, e202501732. - Synthesis of S- and N,S-heterocycles by gold-catalyzed cyclizations
Van Wesemael C., Choury M., Wagner P., Rognan C., Blond G., Gulea M.
Phosphorus, Sulfur Silicon Relat. 2025, 198:6, 532-535 (Special issue 30th International Symposium on Organic Chemistry of Sulfur, ISCO30, proceeding). - LPS2336, a New TREK-1 Channel Activator Identified by High Throughput Screening
Boyer R., Bony R., Maugis M., Schopp J., Leroux M., Michelin C., Gonthier L., Grzeskiewicz Q., Jouannet A., Aissouni Y., Didier B., Gulea M., Girard N., Cintrat J.-C., Dumeige A., Busserolles J., Ducki S., Lolignier S.
Biomolecules 2025, 15, 740. - Orthogonal Tandem Catalysis involving Au(I)-Hydroacyloxylation and Rh(I)-Hydroformylation reactions
Salvi E., Galéa R., Van Wesemael C., Wagner P., Girard N., Blond G.
Org. Chem. Front. 2025, 12, 3050-3057. - Doyle-Kirmse Reaction of S-Allyl and S-Propargyl Phosphorothioates
Tual L., Rognan C., Maujean T., Pertschi R., Girard N., Blond G., Gulea M.
Synthesis 2025, 57, 1490-1498.
2024
- Reduction of S=O and SO2 to S, S-X to S-H and P=O to P.
Magné V., Serusi L., Gulea M., Hanquet G., Madec D., Panossian A.
Comprehensive Organic Synthesis; N. Maulide (volume editor), 3nd edition, Volume 8, 2024. - Domino Doyle-Kirmse/Claisen-Thioimidate Rearrangements: Access to 2-Aminobuta-1,3-diene Derivatives of Benzazole-2-thiones
Rognan C., Locquet P., Pertschi R., Girard N., Gulea M.
Adv. Synth. Catal. 2024, 366, 4078 – 4083. - The IMS Library: From In-Stock to Virtual.
Djikic-Stojsic T., Bret G., Blond G., Girard N., Le Guen C., Marsol C., Schmitt M., Schneider S., Bihel F., Bonnet D., Gulea M., Kellenberger E.
ChemMedChem 2024, 19, e202400381. - Hetero-Diels–Alder and CuAAC Click Reactions for Fluorine-18 Labeling of Peptides: Automation and Comparative Study of the Two Methods.
Maujean T., Ramanoudjame S. M., Riché S., Le Guen C., Boisson F., Muller S., Bonnet D., Gulea M., Marchand P.
Molecules 2024, 29, 3198. - Hydroformylation of Alkynyl Sulfides: A Stereo- and Regioselective Route to alpha-Sulfenyl Acroleins.
Wagner P., Gulea M., Girard N.
Adv. Synth. Catal. 2024, 366, 1298-1305.
2023
- Rapid and Highly Selective Fluorescent Labeling of Peptides via a Thia-Diels-Alder Cycloaddition: Application to Apelin.
Maujean T., Wagner P., Valencia C., Riché S., Iturrioz X., Villa P., Girard N., Karpenko J., Gulea M., Bonnet D.
Bioconjugate Chem. 2023, 34, 1, 162–168 - Catalyst-free thia-Diels-Alder click reaction for the labeling of peptides for imaging applications.
Maujean T., Marchand P., Wagner P., Riché S., Boisson F., Girard N., Karpenko J., Bonnet D., Gulea M.
Phosphorus, Sulfur Silicon Relat. 2023, special issue 29th International Symposium on Organic Chemistry of Sulfur (ISOCS29) - Synthesis of new N/S-containing compounds by Pd-catalyzed tandem reactions
Lopes A. B., Choury M., Wagner P., Gulea M.
Phosphorus, Sulfur Silicon Relat. 2023, special issue 29th International Symposium on Organic Chemistry of Sulfur (ISOCS29)
2022
- Gold(I)-Catalyzed Carbothiolation via Rearrangement of S- Propargyl Group: An Access to 3-Allenyl or 3-Indenyl Benzo[b]thiophenes
Van Wesemael C., Brach N., Gulea M., Blond G.
Adv. Synth. Catal. 2022, 364, 4141–4145 (VIP) - Hetero-Diels-Alder Click Reaction of Dithioesters for a Catalyst-Free Indirect 18F-Radiolabelling of Peptides
Maujean T., Marchand P., Wagner P., Girard N., Riché S., Boisson F., Bonnet D., Gulea M.
Chem. Commun., 2022, 58, 11151-11154 - Access to 1,4-Thiazepanes via Gold-Catalyzed 7-exo-dig Thioallylation and their Cycloisomerization to Bicyclic [4.3.1] Bridgehead-Olefinic Systems
Choury M., Wagner P., Rognan C., Blond G., Gulea M.
Adv. Synth. Catal., 2022, 364, 3238-3244 - Gold(I)-Catalyzed Domino Reaction : An Access to furooxepines
Galéa R., Blond G.
Adv. Synth. Catal., 2022, 364, 1532-1536
2021
- An Alternative Route to Complex Allenes or Cyclooctatrienes via a Suzuki Cyclocarbopalladation Cascade
Flores O., Locquet P., Suffert J.
Chem. Eur. J., 2021, 10.1002/chem.202103502 -
Two-photon sensitive coumarinyl photoremovable protecting groups with rigid electron-rich cycles obtained by domino reactions initiated by a 5-exo-dig cyclocarbopalladation
Chaud J., Morville C., Bolze F., Garnier D., Chassaing S., Blond G., Specht A.
Org. Lett., 2021, 10.1021/acs.orglett.1c02778 - 4-exo-dig Cyclocarbopalladation, Discovery and Application in the Synthesis of Complex Polycyclic Molecules
Blond G., Suffert J.
Strategies and Tactics in Organic Synthesis, Elsevier, 2021, Vol. 15, Chapitre 10 -
Cyclocarbopalladation/Stille Cascade: Stereoselective Access to Quaternary Functionalized Carbons
Flores O., Wagner P., Suffert J.
Org. Lett. 2021, 23, 6568–6572 -
Unravelling the Puzzle of Anthranoid Metabolism in Living Plant Cells Using Spectral Imaging Coupled to Mass Spectrometry
Chevalier Q., Gallé J.-B., Wasser N., Mazan V., Vilette C., Mutterer J., Elustondo M. M., Girard N., Elhabiri M., Schaller H., Hemmerlin A., Vonthron-Sénéchau C.
Metabolites 2021, 11, 571 - Diastereoselective oxidation of menthyl arenesulfenates to sulfinates and access to enantioenriched aryl methyl sulfoxides
Hamel M., Vazeux M., Gulea M.
Chemical Papers, 2021, 75, 6137-6143 - A Synthetic Route to Benzothiazocines with Two or Three Carbon Stereocenters via Copper-Catalyzed Intramolecular N-Arylation
Choury M., Blond G., Gulea M.
Eur. J. Org., 2021, 2203-2211 - 2D and 3D Silver-Based Coordination Polymers with Thiomorpholine-4-carbonitrile and Piperazine-1,4-dicarbonitrile: Structure, Intermolecular Interactions, Photocatalysis, and Thermal Behavior
Ristic P., Filipović N. R., Blagojević V., Ćirković J., Hollo B., Djokic V. R., Donnard M., Gulea M., Marjanović I., Klisurić O. R.,Todorović T. R.
CrystEngComm, 2021, 23, 4799–4815
2020
- Bicyclic 5-5 Systems With One Ring Junction Nitrogen Atom: One Extra Heteroatom 1:0
Suffert J.
Reference Module in Chemistry, Molecular Sciences and Chemical Engineering, Elsevier, 2020 -
Three Cheers for Nitrogen: Aza-DKPs, the Aza Analogues of 2,5-Diketopiperazines
Maujean T., Girard N., Ganesan A., Gulea M., Bonnet D.
RSC Adv., 2020, 10, 43358 -
Endocyclic Enamides Derived from Aza‐Diketopiperazines as Olefin Partners in Povarov Reaction: An Access to Tetracyclic N‐Heterocycles
Maujean T., Chataigner I., Girard N., Gulea M., Bonnet D.
Eur. J. Org. Chem., 2020, 7385-7395 -
Gold(I)-Catalyzed Domino Reaction for Furopyrans Synthesis
Ruch M., Brach N., Galéa R., Wagner P., Blond G.
Molecules, 2020, 25, 4976 -
Solvent Effect in Gold(I)-Catalyzed Domino Reaction: Access to Furopyrans
Wagner P., Ghosh N., Gandon V., Blond G.
Org. Lett., 2020, 22, 18, 7333–7337 -
Synthesis of Medium-Sized Heterocycles by Transition-Metal-Catalyzed Intramolecular Cyclization
Choury M., Basilio Lopes A., Blond G., Gulea M.
Molecules, 2020, 25, 3147 - Sustainable Synthetic Approaches Involving Thiocyanation and Sulfur-Cyanation: An Update
Gulea M. and Donnard M.
Current Green Chemistry, 2020, 7, 201-207 - 1D and 2D Silver-Based Coordination Polymers with Thiomorpholine-4-carbonitrile and Aromatic Polyoxoacids as Coligands: Structure, Photocatalysis, Photoluminescence, and TD- DFT Study
Ristić P., Todorović T. R., Blagojević V., Klisurić O. R., Marjanović I., B. Barta Holló, Vulić P., Gulea M., Donnard M., Monge M., Rodríguez-Castillo M., López-de-Luzuriaga J. M. and Filipović N. R.
Cryst. Growth Des., 2020, 20, 4461–4478 - Influence of C–H/X (X = S, Cl, N, Pt/Pd) Interactions on the Molecular and Crystal Structures of Pt(II) and Pd(II) Complexes with Thiomorpholine-4-carbonitrile: Crystallographic, Thermal, and DFT Study
Ristić P., Blagojević V., Janjić G., Rodić M., Vulić P., Donnard M., Gulea M., Chylewska A., Makowski M., Todorović T., Filipović N.
Cryst. Growth Des., 2020, 20, 3018-3033
2019
- Ligand-Controlled Regiodivergent Hydroformylation of Ynamides: A Stereospecific and Regioselective Access to 2- and 3-Aminoacroleins
Wagner P., Donnard M., Girard N.
Org. Lett., 2019, 10.1021/acs.orglett.9b03566 - Silver-based monomer and coordination polymer with organic thiocyanate ligand: Structural, computational and antiproliferative activity study
Filipović N. R., Ristić P., Janjić G. , Klisurić O., Puerta A., Padrón J. M., Donnard M., Gulea M., Todorović
T. R.
Polyhedron, 2019, 173, 114132 - Gold(I)-Catalyzed Synthesis of Furopyrans: Insight into Hetero-Diels–Alder Reactions
Pertschi R., Wagner P., Ghosh N., Gandon V., Blond, G. - Tandem Double-Cross-Coupling/Hydrothiolation Reaction of 2-Sulfenyl Benzimidazoles with Boronic Acids
- Synthesis of Aromatic Rings Embedded in Polycyclic Scaffolds by Triyne Cycloaddition: Competition between Carbonylative and Non-Carbonylative Pathways
Salacz L., Girard N., Suffert J., Blond G.
Molecules, 2019, 24, 595 (Open Access) - Synthesis of benzimidazole‐fused medium‐sized N,S‐heterocycles via palladium‐catalyzed cyclizations
2018
- Versatile Synthetic Approach for Selective Diversification of Bicyclic Aza-Diketopiperazines
Péron F., Riché S., Lesur B., Hibert M., Breton P., Fourquez J.-M., Girard N., Bonnet D.
ACS Omega, 2018, 3, 15182−15192 -
Progress in the Chemistry of Phosphorothioates
Gulea M.
Advances in Organic Synthesis, Atta-ur-Rahman (Ed.), 2018, 12, 117-150
- Synthesis of Polyheterocyclic Tropones by [2+2+2+1] Carbonylative Cycloaddition of Triynes
Salacz L., Girard N., Blond G., Suffert J.
Org. Lett., 2018, 20, 3915-3918
- Molecular Diversity of Cyclooctatetraenes through Palladium-Catalyzed Cascade Reactions
Blouin S., Pertschi R., Schoenfelder A., Suffert J., Blond G.
Adv. Synth. Catal., 2018, 360, 2166-2171 (VIP) - Synthesis of Sulfur-Containing Exo-Bicyclic Dienes and Their Diels–Alder Reactions To Access Thiacycle-Fused Polycyclic Systems
Castanheiro T., Schoenfelder A., Donnard M., Chataigner I., Gulea M.
J. Org. Chem., 2018, 83, 4505-4515
- Carbonylative cycloadditions for the synthesis of medium-sized carbo- and heterocycles.
Salacz L., Girard N., Suffert J., Blond G.
Monatshefte für Chemie - Chemical Monthly, 2018, 149, 671-686
2017
- Pd and Cu-mediated domino reactions for the synthesis of sulfur heterocycles.
Donnard M., Castanheiro T., Gulea M.
in Targets in Heterocyclic Systems (book chapter), vol. ed. Orazio Attanassi, Perdo Merino et Domenico Spinelli, Societa Chimica Italiana, 2017, vol. 21, 255-276 -
Synthesis of Benzo[c]silole derivatives Bearing a Tetrasubstituted Exocyclic C=C Double Bond by Palladium-Catalyzed Domino Reactions.
Wagner P., Gulea M., Suffert J., Donnard M.
Chem. Eur. J., 2017, 23, 7458-7462 - Intramolecular inverse electron-demand [4+2] cycloadditions of ynamidyl-tethered pyrimidines: comparative studies in trifluorotoluene and sulfolane
Donnard M., Duret G., Bisseret P., Blanchard N.
Comptes Rendus Chimie, 2017, 20, 643-647 (OPEN ACCESS) -
Desymmetrizing Hydroformylation of Dihydromuconic Acid Diesters: Application to the Synthesis of (+/-)-Vindeburnol
Salacz L., Charpentier C., Suffert J., Girard N.
J. Org. Chem., 2017, 82, 2257-2262 - Synthesis of original polycycles containing 5, 6 and 7-membered rings through cyclocarbopalladations/CH-activation cascade reactions.
Joussot J., Schoenfelder A., Suffert J., Blond G.
Comptes Rendus Chimie, 2017, 20, 665-681 (OPEN ACCESS) -
Cyclocarbopalladation as a key step in cascade reactions: recent developments.
Blouin S., Blond G., Donnard M., Gulea M., Suffert J.
Synthesis, 2017, 49, 1767-1784 -
Comparative study on the reactivity of propargyl and alkynyl sulfides in Palladium-catalyzed domino reactions
Castanheiro T., Suffert J., Donnard M., Gulea M.
Comptes Rendus Chimie, 2017, 20, 624-633 (OPEN ACCESS) -
Hopping of Palladium: Access to Original Polycyclic Structures Containing Three-, Four-, Five- and Six-Membered Rings
Ghosh N., Maiereanu C., Suffert J., Blond G.
Synlett, 2017, 28, 451-455 -
Synthesis of Sulfur Heterocycles via Domino Metal-Mediated Reactions
Castanheiro T., Suffert J., Donnard M., Gulea M.
Phosphorus Sulfur Silicon Relat. Elem., 2017, 192, 162 -
Pro-differentiating effects of a synthetic flavagline on human teratocarcinomal cancer stem-like cells.
Emhemmed F., Ali Azouaou S., Zhao Q., Appert-Collin A., Bennasroune A., Schini-Kerth V.B., Muller C.D., Désaubry L., Fuhrmann G.
Cell Biol Toxicol., 2017, ASAP
