Publications

publicationpublibook


2017

  • Synthesis of Benzo[c]silole derivatives Bearing a Tetrasubstituted Exocyclic C=C Double Bond by Palladium-Catalyzed Domino Reactions.
    Wagner P., Gulea M., Suffert J., Donnard M.
    Chem. Eur. J., 2017, 23, 7458-7462

  • Desymmetrizing Hydroformylation of Dihydromuconic Acid Diesters: Application to the Synthesis of (+/-)-Vindeburnol
    Salacz L., Charpentier C., Suffert J., Girard N.
    J. Org. Chem.
    , 2017, 82, 2257-2262

  • Synthesis of original polycycles containing 5, 6 and 7-membered rings through cyclocarbopalladations/CH-activation cascade reactions.
    Joussot J., Schoenfelder A., Suffert J., Blond G.
    Comptes Rendus Chimie, 2017, 20, 665-681 (OPEN ACCESS)
  • Cyclocarbopalladation as a key step in cascade reactions: recent developments.
    Blouin S., Blond G., Donnard M., Gulea M., Suffert J.
    Synthesis, 2017, 49, 1767-1784

  • Comparative study on the reactivity of propargyl and alkynyl sulfides in Palladium-catalyzed domino reactions
    Castanheiro T., Suffert J., Donnard M., Gulea M.
    Comptes Rendus Chimie,
    2017, 20, 624-633 (OPEN ACCESS)

  • Intramolecular inverse electron-demand [4+2] cycloadditions of ynamidyl-tethered pyrimidines: comparative studies in trifluorotoluene and sulfolane
    Donnard M., Duret G., Bisseret P., Blanchard N.
    Comptes Rendus de Chimie, 2017, 20, 643-647  (OPEN ACCESS)

  • Hopping of Palladium: Access to Original Polycyclic Structures Containing Three-, Four-, Five- and Six-Membered Rings
    Ghosh N., Maiereanu C., Suffert J., Blond G.
    Synlett,
    2017, 28, 451-455

  • Synthesis of Sulfur Heterocycles via Domino Metal-Mediated Reactions
    Castanheiro T., Suffert J., Donnard M., Gulea M.
    Phosphorus Sulfur Silicon Relat. Elem., 2017, 192162-165


2016

  • Recent Contributions to Hetero Diels-Alder Reactions
    Blond G., Gulea M., Mamane V.
    Curr. Org. Chem., 2016, 20, 2161
  • A Step-Economical Multicomponent Synthesis of 3D-Shaped Aza-Diketopiperazines and Their Drug-like Chemical Space Analysis
    Regenass P.M.Riché S., Peron F., Rognan D., Hibert M., Girard N., Bonnet D.
    Org. Biomol. Chem.,
    2016, 14, 8859-8863

  • Synthesis of 3-Substituted Chromones and Quinolones from Enaminones
    Joussot J., Schoenfelder A., Larquetoux L., Nicolas M., Suffert J., Blond G.
    Synthesis, 2016, 48, 3364-3372
  • Aerobic Copper-Mediated Domino Three-Component Approach to 2-Aminobenzothiazole Derivatives.
    Castanheiro T., Suffert J., Gulea M., Donnard M.
    Org. Lett.
    , 2016, 18, 2588   (OPEN ACCESS)

  • Synthesis of Cyclooctatetraenes through a Palladium-Catalyzed Cascade Reaction.
    Blouin S., Gandon V., Blond G., Suffert J.
    Angew. Chem. Int. Ed.,
    2016, 55, 7208
  • Hedgehog associated to microparticles inhibits adipocyte differentiation via a non-canonical pathway.
    Fleury A., Hoch L., Martinez MC, Faure H., Taddei M., Petricci E., Manetti F., Girard N., Mann A., Jacques C., Larghero J., Ruat m., Adriantsitohaina R., LeLay S.
    Scientific Reports, 2016, 23479

  • Recent Advances in the Chemistry of Organic Thiocyanates.
    Castanheiro T., Suffert J., Donnard M., Gulea M.
    Chem. Soc. Rev., 2016, 45, 494-505


2015

  • MRT-92 inhibits Hedgehog signaling by blocking overlapping binding sites in the transmembrane domain of the smoothened receptor.

    Hoch, L.; Faure, H.; Roudaut, H.; Schoenfelder, A.; Mann, A.; Girard, N.; Bihannic, L.; Ayrault, O.; Petricci, E.; Taddei, M.
    FASEB 2015, 19, 1817-1829

2014

  • Practical access to aromatic thiocyanates by CuCN-mediated direct aerobic oxidative cyanation of thiophenols and diaryl disulfides.
    Castanheiro, T.;  Gulea, M.; Donnard, M.; Suffert, J.
    Eur. J. Org. Chem., 2014, 2014, 7814-7817.
  • Diastereoselective synthesis of novel aza-diketopiperazines via a domino cyclohydrocarbonylation/addition process.
    Regenass, P.; Margathe, J.-F.; Mann, A.; Suffert, J.; Hibert, M.; Girard, N.; Bonnet, D.
    Chem. Commun. 2014, 50, 9657–9660.

  • Cyclocarbopalladation/cross-coupling cascade reactions in sulfide series: access to sulfur heterocycles.
    Castanheiro, T.; Donnard, M.; Gulea, M.; Suffert, J.
    Org. Lett.
    2014, 16, 3060–3063.

2013

  • Discovery, Molecular and Pharmacological Characterization of GSA-10, a Novel Small-Molecule Positive Modulator of Smoothened
    Tatiana Gorojankina, Lucile Hoch, Hélène Faure, Hermine Roudaut, Elisabeth Traiffort, Angèle Schoenfelder, Nicolas Girard, André Mann, Fabrizio Manetti, Antonio Solinas, Elena Petricci, Maurizio Taddei, and Martial Ruat
    Molecular Pharmacology
    2013, 83, 1020-1029
  • Asymmetric Three-Component Domino Reaction: An Original Access to Chiral Nonracemic 1,3-Thiazin-2-ones
    Flavie Peudru, Fabien Le Cavelier, Jean-Francois Lohier, Mihaela Gulea and Vincent Reboul
    Org. Lett.
    2013, 15, 5710-5713

    Highlighted in SYNFACTS 2014 by Victor Snieckus, Jane Panteleev (Pfizer), 0320014, 10(2), 0136
  • Ortho-(methylsulfanyl)phenylphosphonates and derivatives: Synthesis and applications as mono- or bidentate ligands for the preparation of platinum complexes
    Matthieu Hamela, Mathieu Lecinq, Mihaela Gulea, Jiří Kozelka
    J. Organomet. Chem.
    2013, 745-746, 206-213
  • Expeditious cascade reactions: controlled syntheses of fenestradienes and cyclooctatrienes under palladium catalysis
    Mélanie Charpenay, Aicha Boudhar, Catherine Hulot, Gaëlle Blond, Jean Suffert 
    Tetrahedron
    2013, 69, 7568-7591
    special issue in honour of Pr Paul A. Wender

2012

  • Acylthiourea, acylurea, and acylguanidine derivatives with potent hedgehog inhibiting activity.
    Solinas, A.; Faure, H.; Roudaut, H.; Traiffort, E.; Schoenfelder, A.; Mann, A.; Manetti, F.; Taddei, M.; Ruat, M.
    J. Med. Chem
    .
    2012, 55, 1559–1571.
  • Trimethoxyarene as a Highly Ionizable Tag for Reaction Analysis by Atmospheric Pressure Photoionization Mass Spectrometry (APPI/MS): Exploration of Heterocyclic Synthesis.
    Bui The Thuong, M.; Catala, C.; Colas, C.; Schaeffer, C.; Van Dorsselaer, A.; Mann, A.; Wagner, A.
    Eur. J. Org. Chem. 2012, 85–92

  • Stereoselective Multicomponent Assembly of Enantiopure Oxazolopiperidines and -azepines.
    Zill, N.; Schoenfelder, A.; Girard, N.; Taddei, M.; Mann, A.
    J. Org. Chem.
    2012, 77, 2246-2253

  • Mild chemo-selective hydration of terminal alkynes catalysed by AgSbF6
    Bui The Thuong, M.; Mann, A.; Wagner, A.
    Chem. Commun. 2012, 48, 434-436

2011

  • Cyclohydrocarbonylation-Based Strategy toward Poly- Substituted Piperidines.
    Arena, G.; Zill, N; Salvadori, J.; Girard, N.; Mann, A.; Taddei, M.
    Org. Lett.
    2011, 13, 2294–2297
  • Identification of a low–molecular weight TrkB antagonist with anxiolytic and antidepressant activity in mice
    Cazorla, M.; Prémont, J.; MAnn, A.; Girard, N.; Kellendonk, C.; Rognan, Didier

    J. Clin. Invest. 2011, 121, 1846-1857

  • New Palladium-Catalyzed Cascades: 4-exo-dig Cyclocarbopalladation Reaction Followed by Suzuki-Miyaura or Sonogashira Cross-Coupling
    Charpenay, M.; Boudhar, A.; Siby, A.; Schigand, S.; Blond, G.; Suffert, J.
    Adv. Synth. Catal. 2011, 353, 3151-3156

  • Microwave-Assisted Domino Hydroformylation without Syngas
    Cini, E.; Airiau, E.; Girard, N.; Mann, A.; Salvadori, J.; Taddei, M.
    Synlett 2011, 199-202