Publications


2014

  • Single cell tracking assay reveals an opposite effect of selective small non-peptidic alpha 5 beta 1 or alpha v beta 3/beta 5 integrin antagonists in U87MG glioma cells
    Ray, A.-M.;Schaffner, F.;Janouskova, H.;Noulet, F.;Rognan, D.;Lelong-Rebel, I.;Choulier, L.;Blandin, A.-F.;Lehmann, M.;Martin, S.;Kapp, T.;Neubauer, S.;Rechenmacher, F.;Kessler, H. and Dontenwill, M.
    Biochimica Et Biophysica Acta-General Subjects 2014
    , 1840, 2978-2987
  • Design of a General-Purpose European Compound Screening Library for EU-OPENSCREEN
    Horvath, D.;Lisurek, M.;Rupp, B.;Kuehne, R.;Specker, E.;von Kries, J.;Rognan, D.;Andersson, C. D.;Almqvist, F.;Elofsson, M.;Enqvist, P.-A.;Gustavsson, A.-L.;Remez, N.;Mestres, J.;Marcou, G.;Varnek, A.;Hibert, M.;Quintana, J. and Frank, R.
    Chemmedchem 2014, 9, 2309-2326

2013

  • TRAF4 Is a Novel Phosphoinositide-Binding Protein Modulating Tight Junctions and Favoring Cell Migration
    Rousseau, A.;McEwen, A. G.;Poussin-Courmontagne, P.;Rognan, D.;Nomine, Y.;Rio, M.-C.;Tomasetto, C. and Alpy, F.
    Plos Biology
    2013, 11,
  • Ligand promiscuity or protein redundancy?: Lessons from the PDB
    Kellenberger, E.;Sturm, N.;Desaphy, J. and Rognan, D.
    Abstracts of Papers of the American Chemical Society
    2013, 246,
  • Glucose 6P Binds and Activates HlyIIR to Repress Bacillus cereus Haemolysin hlyII Gene Expression
    Guillemet, E.;Tran, S.-L.;Cadot, C.;Rognan, D.;Lereclus, D. and Ramarao, N.
    Plos One
    2013, 8,
  • Exploration of the Orthosteric/Allosteric Interface in Human M1 Muscarinic Receptors by Bitopic Fluorescent Ligands
    Daval, S. B.;Kellenberger, E.;Bonnet, D.;Utard, V.;Galzi, J.-L. and Ilien, B.
    Molecular Pharmacology
    2013, 84, 71-85
  • Telaprevir: protease inhibitor drug against hepatitis C
    Bourel-Bonnet, L. and Kellenberger, E.
    Virologie
    2013, 17, 3-5

2012

  • Use of an alpha 5 beta 1 Small Non-peptidic Antagonist to Inhibit Glioblastoma Migration Fostered by Integrin Expression
    Ray, A.;Janouskova, H.;Lehmann, M.;Bonnet, D.;Villa, P.;Brino, L.;Martin, S.;Rebel, I. L.;Rognan, D. and Dontenwill, M.
    European Journal of Cancer 2012, 48, S244
  • Selective Fluorescent Nonpeptidic Antagonists For Vasopressin V-2 GPCR: Application To Ligand Screening and Oligomerization Assays
    Loison, S.;Cottet, M.;Orcel, H.;Adihou, H.;Rahmeh, R.;Lamarque, L.;Trinquet, E.;Kellenberger, E.;Hibert, M.;Durroux, T.;Mouillac, B. and Bonnet, D.
    Journal of Medicinal Chemistry 2012, 55, 8588-8602
  • Insights into the Mechanism of Bovine CD38/NAD+Glycohydrolase from the X-Ray Structures of Its Michaelis Complex and Covalently-Trapped Intermediates
    Egea, P. F.;Muller-Steffner, H.;Kuhn, I.;Cakir-Kiefer, C.;Oppenheimer, N. J.;Stroud, R. M.;Kellenberger, E. and Schuber, F.
    Plos One 2012, 7,
  • Fluorescent Derivatives of AC-42 To Probe Bitopic Orthosteric/Allosteric Binding Mechanisms on Muscarinic M1 Receptors
    Daval, S. B.;Valant, C.;Bonnet, D.;Kellenberger, E.;Hibert, M.;Galzi, J.-L. and Ilien, B.
    Journal of Medicinal Chemistry 2012, 55, 2125-2143
  • Stereoselective functionalization of pyrrolidinone moiety towards the synthesis of salinosporamide A
    Barbion, J.;Sorin, G.;Selkti, M.;Kellenberger, E.;Baati, R.;Santoro, S.;Himo, F.;Pancrazi, A.;Lannou, M.-I. and Ardisson, J.
    Tetrahedron 2012, 68, 6504-6512

1987 - 2011

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